Multi-Step Organic Synthesis A Guide Through Experiments by Nicolas Bogliotti (informative book of chemistry)
Free download Multi-Step Organic Synthesis A Guide Through Experiments by Nicolas Bogliotti
Authors of: Multi-Step Organic Synthesis A Guide Through Experiments by Nicolas Bogliotti
Nicolas Bogliotti
Roba Moumne
Table of Contents in Multi-Step Organic Synthesis A Guide Through Experiments by Nicolas Bogliotti
Preface
List of Abbreviations
1 Atovaquone: An Antipneumocystic Agent
Answers
References
2 SEN794: An SMO Receptor Antagonist
Answers
References
3 Synthesis of an H1–H3 Antagonist
3.1 Synthesis of Fragment 2
3.2 Synthesis of Fragment 3
3.3 Fragment Assembly and End of Synthesis
Answers
References
4 Synthesis of Eletriptan
Answers
References
5 Total Synthesis and Structure Revision of Streptophenazine A
Answers
References
6 Synthesis of Leiodermatolide, A Biologically Active Macrolide
6.1 Access to Fragment C
6.1.1 Preparation of Compound 2
6.1.2 Preparation of Compound 7
6.1.3 Preparation of Compound 12
6.1.4 Preparation of Fragment C
6.2 Access to Fragment D
6.2.1 Preparation of Compound 26
6.2.2 Preparation of Fragment D
6.3 Final Steps
6.3.1 Assembly of B and Formation of A by Ring‐Closing Alkyne
Metathesis
6.3.2 Coupling of Sugar and Macrocycle
Answers
References
7 Azobenzene-Thiourea Catalysts for the Control of Chemical Reactivity
with Light
7.1 Synthesis of Azobenzene-Thiourea Derivatives
7.2 Investigation of Catalytic Properties
Answers
References
8 Synthesis and Properties of a Photo-activatable Mimic of Pyridoxal
5ʹ-Phosphate
Answers
References
9 Fluorescent Peptides for Monitoring Activity of Autophagy-Initiating
Enzyme
9.1 Solid-Phase Synthesis of a Putative Fluorogenic Peptide Substrate
for ATG4B
9.2 Evaluation as Fluorogenic Substrates for ATG4B
9.3 Solution-Phase Synthesis of a Fluorogenic Substrate Analog
Containing a Self-Immolating Linker
Answers
References
10 Fluorescent Peptide Probes for Cathepsin B
10.1 Solution Synthesis of a Water-Soluble Cyanine Fluorophore
10.2 Synthesis of a Water-Soluble Cyanine Fluorophore Using a Polymeric
Support
10.3 Synthesis and Evaluation of Cyanine-Based NIR Peptide Probes
for Monitoring Cathepsin B Activity
Answers
References
11 Total Synthesis of Stemoamide
11.1 Radical Approach to the Construction of the Tricyclic Core
of Stemoamide
11.2 Formal Synthesis of (±)-Stemoamide
11.3 Enantioselective Total Synthesis of (−)-Stemoamide
Answers
References
12 Total Synthesis and Structure Revision of Caraphenol B
12.1 Synthesis of the Proposed Structure of Caraphenol B
12.2 Synthesis of the Revised Structure of Caraphenol B
Answers
References
13 Synthetic Routes Toward Muricatacin and Analogs
13.1 Synthesis of (+)-Muricatacin
13.2 Synthesis of (+)-epi-Muricatacin by Enantioselective Ketone
Reduction
13.3 Synthesis of (−)-Muricatacin
Answers
References
14 Asymmetric Synthesis of (−)-Martinellic Acid
14.1 Preliminary Studies: Toward the Formation of a Model Tricyclic
Compound
14.2 Synthesis of an Advanced Intermediate
14.3 Completion of the Synthesis
Answers
References
15 Cyclic Pseudopeptides as Potent Integrin Antagonists
15.1 Conformational Analysis
15.2 Synthesis of Bicyclic Lactam Templates
15.3 Solid Phase Peptide Synthesis
15.4 Pharmacological Study
Answers
References
16 Enantioselective Synthesis of Nonnatural Amino Acids for Incorporation
in Antimicrobial Peptides
16.1 First Generation Mimetics: Synthesis and Biological Evaluation
16.2 Structural Analysis and Mechanism of Action
16.3 Sequence Optimization: Synthesis of Nonnatural Amino Acids
16.3.1 Synthesis of Homophenylalanine (Hfe)
16.3.2 Synthesis of Phenylglycine (Phg)
16.3.3 Synthesis of 4‐Chlorophenylalanine (ClF)
16.3.4 Synthesis of 2‐Naphtylalanine (2‐Nal)
16.3.5 Synthesis of 1‐Naphtylalanine (1‐Nal)
16.3.6 Synthesis of Cyclohexylalanine (Cha)
16.3.7 Synthesis of Norleucine (Nle)
16.3.8 Synthesis of Biphenylalanine (Bip)
Answers
References
Further Reading
Index
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